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INHIBITORS OF GABA METABOLISMMETCALF BW.1979; BIOCHEM. PHARMACOL.; GBR; DA. 1979; VOL. 28; NO 11; PP. 1705-1712; BIBL. 65 REF.Article

RECENT PROGRESS IN THE DESIGN OF SUICIDE ENZYME INHIBITORSMETCALF BW.1981; ANNU. REP. MED. CHEM.; ISSN 0065-7743; USA; DA. 1981; VOL. 16; PP. 289-297; BIBL. 63 REF.Article

SYNTHETIC ACCESS TO ALPHA -SUBSTITUTED PROP-2-YNYLAMINES AND ALPHA -ACETYLENIC AMINO ACIDS VIA THE T-BUTYL N-TRIMETHYLSILYLPROP-2-YNYLCARBAMATE DIANIONMETCALF BW; CASARA P.1979; J. CHEM. SOC., CHEM. COMMUNIC.; GBR; DA. 1979; NO 3; PP. 119-120; BIBL. 5 REF.Article

TRIMETHYLSILYLACETYLENE-N-CARBOETHOXY GLYCINATE DIANION. A GENERAL SYNTHON FOR ALPHA -ACETYLENIC ALPHA -AMINO ACIDS.CASARA P; METCALF BW.1978; TETRAHEDRON LETTERS; G.B.; DA. 1978; NO 18; PP. 1581-1584; BIBL. 10 REF.Article

SYNTHESIS OF BETA ,GAMMA -UNSATURATED AMINO ACIDS AS POTENTIAL CATALYTIC IRREVERSIBLE ENZYME INHIBITORS.METCALF BW; JUND K.1977; TETRAHEDRON LETTERS; G.B.; DA. 1977; NO 41; PP. 3689-3692; BIBL. 8 REF.Article

CATALYTIC INHIBITION OF GAMMA -AMINOBUTYRIC ACID-ALPHA -KETOGLUTARATE TRANSAMINASE OF BACTERIAL ORIGIN BY 4-AMINOHEX-5-YNOIC ACID, A SUBSTRATE ANALOG.JUNG MJ; METCALF BW.1975; BIOCHEM. BIOPHYS. RES. COMMUNIC.; U.S.A.; DA. 1975; VOL. 67; NO 1; PP. 301-306; BIBL. 15 REF.Article

PHENYL TRANS-2-CHLOROVINYL SULPHONE, A VINYL CATION EQUIVALENTMETCALF BW; BONILAVRI E.1978; J. CHEM. SOC., CHEM. COMMUNIC.; GBR; DA. 1978; NO 21; PP. 914-915; BIBL. 9 REF.Article

ENZYME-ACTIVATED IRREVERSIBLE INHIBITION OF RAT AND MOUSE BRAIN 4-AMINOBUTYRIC ACID-ALPHA -KETOGLUTARATE TRANSAMINASE BY 5-FLUORO-4-OXO-PENTANOIC ACIDLIPPERT B; METCALF BW; RESVICK RJ et al.1982; BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS; ISSN 0006-291X; USA; DA. 1982; VOL. 108; NO 1; PP. 146-152; BIBL. 19 REF.Article

CLEAVAGE OF TERT-BUTYLDIMETHYLSILYL ETHERS BY TETRAFLUOROBORATE SALTSMETCALF BW; BURKHART JP; JUND K et al.1980; TETRAHEDRON LETTERS; GBR; DA. 1980; VOL. 21; NO 1; PP. 35-36; BIBL. 9 REF.Article

SYNTHESIS OF 3-KETO-4-DIAZO-5-ALPHA -DIHYDROSTEROIDS AS A POTENTIAL IRREVERSIBLE INHIBITORS OF STEROID 5-ALPHA -REDUCTASEMETCALF BW; JUND K; BURKUART JP et al.1980; TETRAHEDRON LETTERS; GBR; DA. 1980; VOL. 21; NO 1; PP. 15-18; BIBL. 15 REF.Article

A STEREOSPECIFIC TOTAL SYNTHESIS OF RACEMIC 11ALPHA -HYDROXYPROGESTERONE VIA A BIOMIMETIC POLYENE CYCLIZATIONJOHNSON WS; ESCHER S; METCALF BW et al.1976; J. AMER. CHEM. SOC.; U.S.A.; DA. 1976; VOL. 98; NO 4; PP. 1039-1041; BIBL. 18 REF.Article

EFFECT OF 5-HEXYNE-1,4-DIAMINE ON BRAIN 4-AMINO-BUTYRIC ACID METABOLISM IN RATS AND MICEDANZIN C; JUNG MJ; SEILER N et al.1979; BIOCHEM. PHARMACOL.; GBR; DA. 1979; VOL. 28; NO 5; PP. 633-639; BIBL. 21 REF.Article

4 -AMINO-HEX-5-ENOIC ACID, A SELECTIVE CATALYTIC INHIBITOR OF 4-AMINOBUTYRICACID AMINOTRANSFERASE IN MAMMALIAN BRAIN.LIPPERT B; METCALF BW; JUNG MJ et al.1977; EUROP. J. BIOCHEM.; GERM.; DA. 1977; VOL. 74; NO 3; PP. 441-445; BIBL. 21 REF.Article

DECREASE OF POLYAMINE LEVELS IN RAT TISSUES BY 5-HEXYNE-1,4-DIAMINE, AN ENZYME-ACTIVATED IRREVERSIBLE INHIBITOR OF ORNITHINE DECARBOXYLASEDANZIN C; JUNG MJ; METCALF BW et al.1979; BIOCHEM. PHARMACOL.; GBR; DA. 1979; VOL. 28; NO 5; PP. 627-631; BIBL. 26 REF.Article

THE TIME-DEPENDENT INACTIVATION OF AROMATASE BY 17BETA -HYDROXY-10-METHYLTHIOESTRA-1,4-DIEN-3-ONEFLYNN GA; JOHNSTON JO; WRIGHT CL et al.1981; BIOCHEM. BIOPHYS. RES. COMMUN.; ISSN 0006-291X; USA; DA. 1981; VOL. 103; NO 3; PP. 913-918; BIBL. 15 REF.Article

ALPHA -ETHYNYL AND ALPHA -VINYL ANALOGUES OF ORNITHINE AS ENZYME-ACTIVATED INHIBITORS OF MAMMALIAN ORNITHINE DECARBOXYLASEDANZIN C; CASARA P; CLAVERIE N et al.1981; J. MED. CHEM.; ISSN 0022-2623; USA; DA. 1981; VOL. 24; NO 1; PP. 16-20; BIBL. DISSEM.Article

INHIBITION OF TESTOSTERONE 5ALPHA -REDUCTASE BY A PROPOSED ENZYME-ACTIVATED, ACTIVE SITE-DIRECTED INHIBITORBLOHM TR; METCALF BW; LAUGHLIN ME et al.1980; BIOCHEM. BIOPHYS. RES. COMMUNIC.; USA; DA. 1980; VOL. 95; NO 1; PP. 273-280; BIBL. 29 REF.Article

MECHANISM OF THE STEREOSPECIFIC IRREVERSIBLE INHIBITION OF BACTERIAL GLUTAMIC ACID DECARBOXYLASE BY (R)-(-)-4-AMINOHEX-5YNOIC ACID, AN ANALOGUE OF 4-AMINOBUTYRIC ACIDJUNG MJ; METCALF BW; LIPPERT B et al.1978; BIOCHEMISTRY; USA; DA. 1978; VOL. 17; NO 13; PP. 2628-2632; BIBL. 22 REF.Article

GAMMA -VINYL GABA (4-AMINO-HEX-5-ENOIC ACID), A NEW SELECTIVE IRREVERSIBLE INHIBITOR OF GABA-T: EFFECTS ON BRAIN GABA METABOLISM IN MICE.JUNG MJ; LIPPERT B; METCALF BW et al.1977; J. NEUROCHEM.; G.B.; DA. 1977; VOL. 29; NO 5; PP. 797-802; BIBL. 19 REF.Article

THE EFFECT OF 4-AMINO HEX-5-YNOIC ACID (GAMMA -ACETYLENIC GABA, GAMMA -ETHYNYL GABA) A CATALYTIC INHIBITOR OF GABA TRANSAMINASE, ON BRAIN GABA METABOLISM IN VIVO.JUNG MJ; LIPPERT B; METCALF BW et al.1977; J. NEUROCHEM.; G.B.; DA. 1977; VOL. 28; NO 4; PP. 717-723; BIBL. 35 REF.Article

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